Gold Nanoparticles in Cancer Treatment.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00810
Selective Cytotoxicity to HER2 Positive Breast Cancer Cells by Saporin-Loaded Nanobody-Targeted Polymeric Nanoparticles in Combination with Photochemical Internalization
来源期刊:Molecular PharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01318
Lipolysis-Permeation Setup for Simultaneous Study of Digestion and Absorption in Vitro
来源期刊:Molecular PharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00811
Cell Permeable NBD Peptide-Modified Liposomes by Hyaluronic Acid Coating for the Synergistic Targeted Therapy of Metastatic Inflammatory Breast Cancer.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01123
Synthesis of CSK-DEX-PLGA Nanoparticles for the Oral Delivery of Exenatide to Improve Its Mucus Penetration and Intestinal Absorption.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00809
Novel Hydrogel-Forming Microneedle Array for Intradermal Vaccination in Mice Using Ovalbumin as a Model Protein Antigen.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00895
An Integrated Transfer Learning and Multitask Learning Approach for Pharmacokinetic Parameter Prediction
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00816
Nanoparticle-Induced Controlled Drug Delivery Using Chitosan-Based Hydrogel and Scaffold: Application to Bone Regeneration.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00995
Radioiodinated Portable Albumin Binder as a Versatile Agent for in Vivo Imaging with Single-Photon Emission Computed Tomography.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01116
Electrospinning Optimization of Eudragit E PO with and without Chlorpheniramine Maleate Using a Design of Experiment Approach
来源期刊:Molecular PharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00159
Rational design of PLGA nanoparticles vaccine delivery systems to improve immune responses.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00860
Sulfonamide-Derived Four-Component Molecular Hybrids as Novel DNA-Targeting Membrane Active Potentiators against Clinical Escherichia coli.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01021
In vitro and in vivo behavior of liposomes decorated with PEGs with different chemical features.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00887
Synthesis and Aggregation of a Porphyrin-Cored Hyperbranched Polyglycidol and Its Application as a Macromolecular Photosensitizer for Photodynamic Therapy.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01119
Near-Infrared Fluorescent Peptides with High Tumor Selectivity: Novel Probes for Image-Guided Surgical Resection of Orthotopic Glioma.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00888
Multifunctional Nanocomposites Based on Liposomes and Layered Double Hydroxides Conjugated with Glycylsarcosine for Efficient Topical Drug Delivery to the Posterior Segment of the Eye.
来源期刊:Molecular pharmaceuticsDOI:10.1021/ACS.MOLPHARMACEUT.8B01136
Mechanism of Supersaturation Suppression in Dissolution Process of Acidic Drug Salt.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00006
Host-Guest Interactions between Candesartan and Its Prodrug Candesartan Cilexetil in Complex with 2-Hydroxypropyl-β-cyclodextrin: On the Biological Potency for Angiotensin II Antagonism.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01212
Paclitaxel-Loaded Folate-Coated pH-Sensitive Liposomes Enhance Cellular Uptake and Antitumor Activity.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00329
Nanoconfinement Effects on the Glass Transition and Crystallization Behaviors of Nifedipine.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01172
In Situ Characterization of the Microstructural Evolution of Biopharmaceutical Solid-State Formulations with Implications for Protein Stability.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00935
Targeted Lipid Nanoemulsions Encapsulating Epigenetic Drugs Exhibit Selective Cytotoxicity on CDH1-/FOXM1+ Triple Negative Breast Cancer Cells.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01065
Measuring the pancreatic beta cell mass in vivo with exendin SPECT during hyperglycemia and severe insulitis.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00728
Interplay of supersaturation and solubilization: Lack of correlation between concentration-based supersaturation measurements and membrane transport rates in simulated and aspirated human fluids.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00956
Combination Chemotherapy of L1210 Tumors in Mice with Pretubulysin and Methotrexate Lipo-Oligomer Nanoparticles.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00038
A New Methodology to Create Polymeric Nanocarriers Containing Hydrophilic Low Molecular-Weight Drugs: A Green Strategy Providing a Very High Drug Loading.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00097
Quantitative Imaging of the Hypoxia-Related Marker CAIX in Head and Neck Squamous Cell Carcinoma Xenograft Models
来源期刊:Molecular PharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00950
Detecting functional and accessible folate receptor expression in cancer and polycystic kidneys.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00624
111In-Labeled Glycoprotein Nonmetastatic b (GPNMB) Targeted Gemini Surfactant-Based Nanoparticles against Melanoma: In Vitro Characterization and in Vivo Evaluation in Melanoma Mouse Xenograft Model.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00831
Enhanced Reactive Oxygen Species Levels by Active Benzothiazole Complex mediated Fenton Reaction for Highly Effective Anti-tumor Therapy.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00819
Bifunctional Fusion Proteins Derived from Tumstatin and 4-1BBL for Targeted Cancer Therapy.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01190
Revealing Intermolecular Hydrogen Bonding Structure and Dynamics in a Deep Eutectic Pharmaceutical by Magic-Angle Spinning NMR Spectroscopy
来源期刊:Molecular PharmaceuticsDOI:10.1021/acs.molpharmaceut.9b01075
Impact of a Single Hydrogen Substitution by Fluorine on the Molecular Interaction and Miscibility between Sorafenib and Polymers.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b00970
Lung Tissue Delivery of Virus-Like Particles Mediated by Macrolide Antibiotics.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00180
Hydrophilic Small Molecules That Harness Transthyretin To Enhance the Safety and Efficacy of Targeted Chemotherapeutic Agents.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00432
Incorporation of complexation into coamorphous system dramatically enhances dissolution and eliminates gelation of amorphous lurasidone hydrochloride.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00772
Inhibiting hypoxia and chemotherapy-induced cancer cell metastasis under valid therapeutic effect by an assistance of biomimetic oxygen delivery.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00663
Enhanced oral bioavailability of 2-(phosphonomethyl)-pentanedioic acid (2-PMPA) from its (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (ODOL) based prodrugs.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00637
A Novel Conjugate of Bis[((4-Bromophenyl)amino)quinazoline], a EGFR-TK Ligand, with a Fluorescent Ru(II)-Bipyridine Complex, Exhibits Specific Subcellular Localization in Mitochondria.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00608
Geometry of a TLR2-Agonist-Based Adjuvant Can Affect the Resulting Antigen-Specific Immune Response.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00026
Exendin-4 derivatives with an albumin-binding moiety show decreased renal retention and improved GLP-1 receptor targeting.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00271
Renal Excretion of Dabigatran: The Potential Role of Multidrug and Toxin Extrusion (MATE) Proteins.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00472
Development of Arginine Anchored Nano-Globule with Retrograde Trafficking Inhibitor (Retro-2) for the Treatment of Enterohemorrhagic Escherichia coli outbreak.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00727
Vitamin E-conjugated phosphopeptide inhibitor of the polo-box domain of polo-like kinase 1.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00757
Effect of a Common Genetic Variant (p.V444A) in the Bile Salt Export Pump on the Inhibition of Bile Acid Transport by Cholestatic Medications.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.8b01124
Optimizing lysosomal activation of antibody-drug conjugates (ADCs) by incorporation of novel cleavable dipeptide linkers.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00696
In situ Crystal Growth Rate Distributions of Active Pharmaceutical Ingredients.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00937
Investigations of albumin-insulin detemir complexes using molecular dynamics simulations and free energy calculations.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00839
Development of a Liposomal Formulation of Acetyltanshinone IIA for Breast Cancer Therapy.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00493
MRI Assessment of Prostate-Specific Membrane Antigen (PSMA) Targeting by a PSMA-Targeted Magnetic Nanoparticle: Potential for Image-Guided Therapy.
来源期刊:Molecular pharmaceuticsDOI:10.1021/acs.molpharmaceut.9b00036