Aminopyrazole‐substituted metallophthalocyanines: Preparation, aggregation behavior, and investigation of metabolic enzymes inhibition properties
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800292
Synthesis, characterization, biological evaluation, and molecular docking studies of some piperonyl‐based 4‐thiazolidinone derivatives
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900304
Synthesis and antimicrobial activity of novel 1,2,3‐triazole‐conjugates of quinazolin‐4‐ones
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800302
Interconnection of sulfides and sulfoxides in medicinal chemistry
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800248
Quinolone derivatives: Potential anti‐HIV agent—development and application
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900045
New 2,4‐disubstituted‐2‐thiopyrimidines as VEGFR‐2 inhibitors: Design, synthesis, and biological evaluation
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900089
Synthesis and biological evaluation of novel benzo[c]acridine‐diones as potential anticancer agents and tubulin polymerization inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800307
Design, synthesis, biological evaluation, and molecular modeling studies of rhodanine derivatives as pancreatic lipase inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900029
Novel quinoline derivatives carrying nitrones/oximes nitric oxide donors: Design, synthesis, antiproliferative and caspase‐3 activation activities
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800270
Artemisinin‐derived dimers as potential anticancer agents: Current developments, action mechanisms, and structure–activity relationships
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900240
Design, synthesis, and biological evaluation of new pyrazino[1,2‐a]benzimidazole derivatives as selective cyclooxygenase (COX‐2) inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800265
Design and synthesis of 1,2,4‐triazolo[1,5‐a]pyrimidine derivatives as PDE 4B inhibitors endowed with bronchodilator activity
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900002
Synthesis and anti‐coronavirus activity of a series of 1‐thia‐4‐azaspiro[4.5]decan‐3‐one derivatives
来源期刊:Archiv Der PharmazieDOI:10.1002/ardp.201800330
1H‐1,2,3‐Triazole tethered isatin‐moxifloxacin: Design, synthesis and in vitro anti‐mycobacterial evaluation
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900040
Synthesis of novel gefitinib‐based derivatives and their anticancer activity
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800381
Pharmacological explorations of eco‐friendly amide substituted (Z)‐β‐enaminones as anti‐breast cancer drugs
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800244
Safran
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.18782120438
Synthesis and biological evaluation of sphingosine kinase 2 inhibitors with anti‐inflammatory activity
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800298
Identification of dehydroxy isoquine and isotebuquine as promising antileishmanial agents
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800281
1,2,4‐Triazole‐conjugated 1,3,4‐thiadiazole hybrid scaffolds: A potent ameliorant of carrageenan‐induced inflammation by lessening proinflammatory mediators
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900233
Densely substituted piperidines as a new class of elastase inhibitors: Synthesis and molecular modeling studies
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900061
Identification of new NIK inhibitors by discriminatory analysis‐based molecular docking and biological evaluation
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800374
Synthesis, molecular docking studies, and biological evaluation of novel alkyl bis(4‐amino‐5‐cyanopyrimidine) derivatives
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900027
Discovery to solve multidrug resistance: Design, synthesis, and biological evaluation of novel agents
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900127
Microwave‐assisted synthesis of 1‐substituted‐1H‐benzimidazolium salts: Non‐competitive inhibition of human carbonic anhydrase I and II
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800325
Antileismanial activity, mechanism of action study and molecular docking of 1,4‐bis(substituted benzalhydrazino)phthalazines
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800299
Novel calcitriol analogue with an oxolane group: In vitro, in vivo, and in silico studies
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800315
Design, synthesis, and molecular docking studies of novel pyrazolyl 2‐aminopyrimidine derivatives as HSP90 inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900063
Efficient synthesis of meso‐substituted porphyrins and molecular docking as potential new antioxidant and cytotoxicity agents
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800221
Synthesis, antibacterial evaluation, and DNA gyrase inhibition profile of some new quinoline hybrids
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900086
Chemical structure modifications and nano‐technology applications for improving ADME‐Tox properties, a review
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800213
Enantioselective synthesis and biological investigation of tetrahydro‐β‐carboline‐based HDAC6 inhibitors with improved solubility
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900026
G protein‐coupled receptor binding and pharmacological evaluation of indole‐derived thiourea compounds
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900218
Design, synthesis and biological evaluation of 6‐substituted quinolines derived from cabozantinib as c‐Met inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900101
Synthesis and antiageing properties of antioxidant pseudopeptides designed based on the bioisostere principle
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800354
Quinolone derivatives and their antifungal activities: An overview
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800382
Novel N‐(1‐thia‐4‐azaspiro[4.5]decan‐4‐yl)carboxamide derivatives as potent and selective influenza virus fusion inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900028
Synthesis, docking studies, and pharmacological evaluation of 5HT2C ligands containing the N′‐cyanoisonicotinamidine or N′‐cyanopicolinamidine nucleus
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800373
Bi‐heterocyclic benzamides as alkaline phosphatase inhibitors: Mechanistic comprehensions through kinetics and computational approaches
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800278
Novel ketoprofen–antioxidants mutual codrugs as safer nonsteroidal anti‐inflammatory drugs: Synthesis, kinetic and pharmacological evaluation
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800339
Synthesis and mycobacterial evaluation of 5‐substituted‐6‐acetyl‐2‐amino‐7‐methyl‐5,8‐dihydropyrido‐[2,3‐d]pyrimidin‐4(3H)‐one derivatives
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900068
Design and synthesis of imidazolidinone derivatives as potent anti‐leishmanial agents by bioisosterism
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800290
Discovery and biological evaluation of novel G protein‐coupled receptor 119 agonists for type 2 diabetes
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800267
Exploration of the structure–activity relationship and druggability of novel oxazolidinone‐based compounds as Gram‐negative antibacterial agents
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900129
Sulfonylpiperazines based on a flavone as antioxidant and cytotoxic agents
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900051
Synthesis and biological evaluation of heteroalicyclic cyanoguanidines at histamine receptors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900107
Bioassay of ferulic acid derivatives as influenza neuraminidase inhibitors
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900174
Identification of novel selective Mtb‐DHFR inhibitors as antitubercular agents through structure‐based computational techniques
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201900287
Jod.
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.18270210339
Targeting HIV‐TB coinfection by developing novel piperidin‐4‐substituted imines: Design, synthesis, in vitro and in silico studies
来源期刊:Archiv der PharmazieDOI:10.1002/ardp.201800358